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Antiamoebic Drugs

 Antiamoebic Drugs

1. Intestinal and extraintestinal amoebiasis (Hepatic amoebiasis)

2. Drug effective only intestinal amoebiasis (Luminal amoebiasis)

3. Drug used in  entraintestinal amoebiasis 


1. Intestinal and extraintestinal amoebiasis (Hepatic amoebiasis)

Metronidazole

Tinidazole

Orindazole

Secnidazole

Satranidazole

Emetine

Dehydroemetin



2. Drug effective only intestinal amoebiasis (Luminal amoebiasis)

Diloxanide furoate

Tetracycline

Paromomycin

Quinidochlor

Isoquinoline


3. Drug used in  entraintestinal amoebiasis 

Chloroquine


9. Antimalarials Drug

Classification of antimalarials drug

1. Causal prophylactic (primary tissue schizontocides)

(Destroy parasite in liver cells and prevent invasion of Erythrocytes)

Primaquine 

Pyrimethamine (folate antagonists)



2. (Suppressive form) Blood schizontocides (destroy parasite in RBC and terminal clinical attacks of malaria)

Chloroquine

Quinine

Mefoquine

Halofantrine

Hydroxychloroquinine

Pyrimethamine

Chloroguanide

Artemisinin


3. Tissue schizontocides (act on hypnozoites of P. vivax and P. ovale that reproduce relapse)

Primaquine (Hypnozoitocidal drug)


4. Gametocidal Drug (destroy gametocytes and prevent transmission)

Primaquine

Chloroquine

Quinin



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