Types of Cardiovascular Drugs
1. Anti Anginal Drug
Classification of Anti-Anginal Drug
1. Nitrates
1. Short acting drug
Nitroglycerin or glyceryltrinitate (GTN)
2. Long acting drugs
Isosorbididinitrate
Isosorbidemononitrate
2. Beta-blockers
Atenolol
Propranolol
Metroprolol
Esmolol
3. Calcium (ca2+) channel blocker
1. Phenyl alkylamine
Verapamil
2. Benzothiazepine
Diltiazem
3. Dihydropyridines
Nifedipine
Nimodipine
Felodipine
Amlodipine
Nitrendipine
Lacidipine
Benidipine
4. Potassium (k+) channel opner
Nicorandil
5. Others
Aspirin
Dipyridamole
Ranolazime
2. Anti hypertensive drugs
Classification of antihypertensive drug
1. Diuretics
a. Thiazide diuretics
Indapamide
Chlorothiazide
Hydrochlorothiazide
b. High ceiling diuretics
Furosemide
c. Potassium sparing diuretics
Amiloride
Spironolactone
2. Drug acting on Renin- Angiotensin system
a. Angiotensin converting enzyme inhibitors (ACE inhibitors)
Captopril
Enalapril
Lisinopril
Ramipril
Fosinopril
Benazepril
b. Angiotensin ll receptor antagonist
Losartan
Candesartan
Valsartan
Omlesartan
c. Renin- inhibitors aliskiren
3. Sympatholytics
a. Centrally acting drugs
Clonidine
Methyldopa
b. Adrenergic receptor blockers
I. Alpha - blockers
Prazosin
Terazosin
Doxazosin
Il. Beta-blockers
Propranolol
Atenolol
Ill. Alpha and Beta blockers
Labetalol
4. Calcium channel blockers
Verapamil
Nifedipine
Nicardipine
Nimodipine
Amlodipine
5. Dilators
a. Arteriolar dilators
Hydralazine
Minoxidil
Diazoxide
b. Vasodilators
Gasious vasodilators; Nitric oxide
Nitroglycerin
c. Arteriolar and venular dilators
Sodium nitroprusside
3. Anti- Arrhythmic Drugs
Classification of anti- Arrhythmic Drugs
1. Membrane stabilization Agents; Sodium (Na+) channel blockers
Quinidine
Procainamide
Lingnocaine
2. Anti - andrenergic agents
Beta blockers;
Propranolol
Esmolol
3. Agents widening AP action- potential;
Pottassium channel blockers;
Amiodarone
Ibutilide
Dofetilide
Sotalol
4. Calcium channel blocker
Verapamil
Diltiazem
5. Miscellaneous drugs
Digoxin; use for treatment for paroxysmal supraventricular tachycardia (PSVT)
Atropine; effective in the treatment of ventricular arrhythmias
4. Cardiotonics Drug
a. Cardiac glycosides
Digitoxin
Digoxin
Digitalis
b. Arjuna Bark
5. Lipid lowering Agents/ Hypolipidemic drugs/ Anti-hyperlipidemic drug
1. HMG COA reductase inhibitors (statins)
Lovastatin
Roscivastatin
Atorvastatin
Cerivastatin
Simvastatin
Pravastain
Pitavastain
2. Fibric acids
Gemfibrozil
Clofibrate
Fenofibrate
Cholestopol
Cholesevelam
3. Bile acid binding resins
Cholestyramine
Colestipol
4. Anti oxident
Probucol
5. Miscellaneous
Nicotinic acid
Neomycin
6. Sterol absorption
Ezetimibe
Drug use in Blood Disorder
1. Drug used in Coagulation
a. Vitamin K
1. Vitamin K1; Phylloquinon (derived from plant)
Phytonadione
2. Vitamin K2; Menaquinone (produce in gut by bacteria)
3. Vitamin K3; Menadione (synthetic form)
Converted into Vitamin K2 in liver
Fat soluble;
Menadione
Acetomenadione
Water soluble;
Menadione
Sodium bisulfite
b. Miscellaneous drugs
Fibrinogen (factor l); obtain from human
Antihaemophilic factors (factor Vlll) essential blood clotting protein
Adrenochrome monosemicarbazone
Rutin
c. Antifibrinolytic drugs
2. Anti coagulants Drugs
Classification of anticoagulant drug
1. Parenteral anticoagulants drugs
1. Indirect thrombininhibitors
Heparin
Low molecular weight heparin; Enoxaparin
Dalteparin
Reviparin
Fondaparinux
a. Heparinoids
Heparan sulfate
Dextran sulphate
2. Parenteral DTls (direct thrombin inhibitors)
Hirudin
Lepirudin
Argatroban
2. Oral anticoagulants drugs
a. Coumarin derivatives
Warfarin
Nicoumalone
b. Factor Xa inhibitors
Rivaroxaban
c. Oral DTIs
Dabigatran
3. Fibrinolytic drugs/ thrombolytic drug/Antithrombotic drugs
Streptokinase
Urokinase
4. Antiplatelet drugs
Aspirin
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